Keywords

• 30123-17-2 in stock
• 30123-17-2 On Sale
• Linocaine hydrochloride salt Hot Sale

Quick Details

• ProName: 30123-17-2 in stock 30123-17-2 On Sale...
• CasNo: 30123-17-2
• Molecular Formula: C21H24ClN2NaO4S
• Appearance: Powder
• Application: Used in Pharmaceutical, health food, c...
• DeliveryTime: 3-10days
• PackAge: 100g/pack,1kg/pack,25kg/drum
• Port: Shanghai Port
• ProductionCapacity: 10000 Metric Ton/Month
• Purity: 98%,99%
• Storage: Storage in a dry, ventilated place und...
• Transportation: By Air,EMS,FEDEX,UPS and Special Line
• LimitNum: 1 Kilogram
• Grade: Pharma Grade
• Related Substances: qualified
• Residue on Ignition: qualified
• Heavy Metal: qualified
• Valid Period: 2years
• Batch: 20210720

Superiority

30123-17-2 in stock 30123-17-2 On Sale Linocaine hydrochloride  salt Hot Sale

NMDA receptors) and release of BDNF, in turn affecting neural plasticity. Tianeptine (Stablon) is a novel antidepressant and anxiolytic used to treat depression in Europe. Tianeptine binds mu-opioid receptors in the brain which may give it an advantage over typical antidepressants. Structurally, Tianeptine is a tricyclic antidepressant (TCA), though it`s mechanism of action and side effect profile is unlike other TCAs. Tianeptine is an atypical antidepressant with diverse actions, most notably on the glutamatergic system.1, 2 It attenuates glutamate release and modulates the function of the AMPA receptor.2, 3 Tianeptine also acts as an agonist of the µ-opioid receptor (EC50s = 194 and 641 nM for human and mouse receptors, respectively).4 It is as effective as fluoxetine

White to pale yellow solid. Soluble in DMSO (20mg/ml), DMF (30mg/ml), ethanol (10mg/ml) and water (10mg/ml). Chemical. CAS: 30123-17-2. Formula: C21H24ClN2O4S . Na. MW: 435.9 . 23.0. Synthetic. Tianeptine is an atypical antidepressant with diverse actions, most notably on the glutamatergic system. It is a selective facilitator of 5-HT (serotonin) uptake in vitro and in vivo. It attenuates glutamate release and modulates the function of the AMPA receptor. Tianeptine also acts as an agonist of the µ-opioid receptor (EC50s = 194 and 641nM for human and mouse receptors, respectively). Might have anti-inflammatory properties through modulation of TLR and NLRP3 inflammasome signaling pathways.

Details

Synonym: Tianeptine; brand names Stablon, Coaxil, Tatinol, Tianeurax and Salymbra

IUPAC/Chemical Name: sodium 7-((3-chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino)heptanoate

InChi Key: ZLBSUOGMZDXYKE-UHFFFAOYSA-M

InChi Code: InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);/q;+1/p-1

SMILES Code: O=C([O-])CCCCCCNC(C1=CC=C(Cl)C=C12)C3=CC=CC=C3N(C)S2(=O)=O.[Na+]

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001