Keywords

• 30123-17-2 factory sells
• 30123-17-2 superior manufacturer
• Linocaine hydrochloride salt in stock

Quick Details

• ProName: 30123-17-2 factory sells 30123-17-2 su...
• CasNo: 30123-17-2
• Molecular Formula: C21H24ClN2NaO4S
• Appearance: Powder
• Application: Used in Pharmaceutical, health food, c...
• DeliveryTime: 3-10days
• PackAge: 100g/pack,1kg/pack,25kg/drum
• Port: Shanghai Port
• ProductionCapacity: 10000 Metric Ton/Month
• Purity: 98%,99%
• Storage: Storage in a dry, ventilated place und...
• Transportation: By Air,EMS,FEDEX,UPS and Special Line
• LimitNum: 1 Kilogram
• Grade: Pharma Grade
• Related Substances: qualified
• Residue on Ignition: qualified
• Heavy Metal: qualified
• Valid Period: 2years
• Batch: 20210720

Superiority

 factory sells 30123-17-2 superior manufacturer Linocaine hydrochloride  salt in stock

Tianeptine is a drug used primarily in the treatment of major depressive disorder, although it may also be used to treat asthma or irritable bowel syndrome. Chemically it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity (i.e., AMPA receptors and NMDA receptors) and release of BDNF, in turn affecting neural plasticity.

Tianeptine is a tricyclic antidepressant that enhances serotonin uptake. This drug can affect neuroprotection, neuronal excitability, memory and anxiety. However, tianeptine is not linked to adverse psychomotor, cognitive, cardiovascular, sleep and bodyweight effects. The drug has a low tendency for abuse and has a positive pharmacokinetic profile.
Tianeptine is least involved in drug interaction as it is not metabolized by cytochrome P450 system in the liver. In hippocampus and amygdala, tianeptine is involved in glutamatergic transmission processes and elicits neuroplasticity.

Details

• Tianeptine sodium salt

• Short description

  Selective 5-HT uptake enhancer

• Biological description

  Selective 5-HT uptake enhancer. Modulates glutamergic transmission and shows neuroprotective and antidepressant effects. Also shows activity at µ-opioid receptor agonist (K_i = 383 nM). Active in vitro and in vivo.

• Biological action

  Activator

• Purity

  >98%

Properties

• Chemical name

  7-[(3-Chloro-6,11-dihydro-6-methyl- 5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino] heptanoic acid sodium salt

• Molecular Weight

  458.93

• Chemical structure

  

• Molecular Formula

  C₂₁H₂₄ClN₂NaO₄S

• CAS Number

  30123-17-2

• PubChem identifier

  23663953

• SMILES

  CN1C2=CC=CC=C2C(C3=C(S1(=O)=O)C=C(C=C3)Cl)NCCCCCCC(=O)[O-].[Na+]

• InChi

  InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);/q;+1/p-1

• InChiKey

  ZLBSUOGMZDXYKE-UHFFFAOYSA-M

• MDL number

  MFCD00879851

• Appearance

  White solid