Keywords

• 30123-17-2 Hot Sale
• 30123-17-2 Good Supplier In China
• Linocaine hydrochloride salt for sale

Quick Details

• ProName: 30123-17-2 Hot Sale 30123-17-2 Good Su...
• CasNo: 30123-17-2
• Molecular Formula: C21H24ClN2NaO4S
• Appearance: Powder
• Application: Used in Pharmaceutical, health food, c...
• DeliveryTime: 3-10days
• PackAge: 100g/pack,1kg/pack,25kg/drum
• Port: Shanghai Port
• ProductionCapacity: 10000 Metric Ton/Month
• Purity: 98%,99%
• Storage: Storage in a dry, ventilated place und...
• Transportation: By Air,EMS,FEDEX,UPS and Special Line
• LimitNum: 1 Kilogram
• Grade: Pharma Grade
• Related Substances: qualified
• Residue on Ignition: qualified
• Heavy Metal: qualified
• Valid Period: 2years
• Batch: 20210720

Superiority

30123-17-2 Hot Sale 30123-17-2 Good Supplier In China Linocaine hydrochloride  salt for sale

Tianeptine is a drug used primarily in the treatment of major depressive disorder, although it may also be used to treat asthma or irritable bowel syndrome. Chemically it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity 

Tianeptine (sodium salt) is supplied as a crystalline solid. A stock solution may be made by dissolving the tianeptine (sodium salt) in the solvent of choice. Tianeptine (sodium salt) is soluble in organic solvents such as ethanol, DMSO, and dimethyl formamide, which should be purged with an inert gas. The solubility of tianeptine (sodium salt) in these solvents is approximately 10, 20, and 30 mg/ml, respectively. Further dilutions of the stock solution into aqueous buffers or isotonic saline should be made prior to performing biological experiments. Ensure that the residual amount of organic solvent is insignificant, since organic solvents may have physiological effects at low concentrations. Organic solvent-free aqueous solutions of tianeptine (sodium salt) can be prepared by directly dissolving the crystalline solid in aqueous buffers. The solubility of tianeptine (sodium salt) in PBS, pH 7.2, is approximately 10 mg/ml. We do not recommend storing the aqueous solution for more than one day.

Details

• Tianeptine sodium salt

• Short description

  Selective 5-HT uptake enhancer

• Biological description

  Selective 5-HT uptake enhancer. Modulates glutamergic transmission and shows neuroprotective and antidepressant effects. Also shows activity at µ-opioid receptor agonist (K_i = 383 nM). Active in vitro and in vivo.

• Biological action

  Activator

• Purity

  >98%

Properties

• Chemical name

  7-[(3-Chloro-6,11-dihydro-6-methyl- 5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino] heptanoic acid sodium salt

• Molecular Weight

  458.93

• Chemical structure

  

• Molecular Formula

  C₂₁H₂₄ClN₂NaO₄S

• CAS Number

  30123-17-2

• PubChem identifier

  23663953

• SMILES

  CN1C2=CC=CC=C2C(C3=C(S1(=O)=O)C=C(C=C3)Cl)NCCCCCCC(=O)[O-].[Na+]

• InChi

  InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);/q;+1/p-1

• InChiKey

  ZLBSUOGMZDXYKE-UHFFFAOYSA-M

• MDL number

  MFCD00879851

• Appearance

  White solid